79
19
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5036 |
cangrelor tetrasodium
|
GPR; P2Y Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Cangrelor tetrasodium 是三磷酸腺苷类似物,是可逆的选择性血小板P2Y12拮抗剂,也是非特异性的GPR17拮抗剂。它直接阻断腺苷二磷酸诱导的血小板活化和聚集,具有迅速有效的抗血小板作用。 | |||
T5460 |
Mofezolac
莫苯唑酸,莫非佐酸 |
COX | Immunology/Inflammation; Neuroscience |
Mofezolac 是一种非甾体类抗炎药,可缓解疼痛并具有抗炎活性,抑制 COX-1和COX-2的IC50为 1.44 和 447 nM。 | |||
T6594 |
MNS
|
Syk; Src; p97 | Angiogenesis; Tyrosine Kinase/Adaptors; Ubiquitination |
MNS 是一种酪氨酸激酶抑制剂和广谱抗血小板药物,是一种 β-硝基苯乙烯衍生物。它完全抑制 U46619 (IC50:2.1 μM)、ADP (IC50:4.1 μM)、花生四烯酸 (IC50:5.8 μM)、胶原 (IC50:7.0 μM)和凝血酶 (IC50:12.7 μM)诱导的血小板聚集,并抑制 Src (IC50:27.3 μM)、Syk (IC50:2.8 μM) 和 FAK (IC50:97.6 μM)。 | |||
T2629 |
UNC2881
|
TAM Receptor | Tyrosine Kinase/Adaptors |
UNC2881 是一种特异性Mer 激酶抑制剂,可抑制稳态的Mer 激酶磷酸化,其IC50=22 nM。 | |||
T15031 |
CYM50260
|
Others; LPL Receptor | GPCR/G Protein; Others |
CYM50260 是有效的、强选择性的鞘氨醇-1-磷酸 4 受体 (S1P4-R) 激动剂 (EC50= 45 nM),对 S1P1-R,S1P2-R,S1P3-R 和 S1P5-R 无活性。 | |||
T6236 |
Ozagrel
奥扎格雷,OKY-046,Domenan |
Thrombin; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Proteases/Proteasome |
Ozagrel (Domenan) 是血栓烷 A2(TXA2) 合酶抑制剂,可抑制哮喘。它也是一种抗血小板剂,可选择性抑制人血小板聚集,IC50为 53.12 μM。 | |||
T15047 |
Dacisteine
N,S-Diacetyl-L-cysteine,达西司坦 |
Others | Others |
Dacisteine (N,S-Diacetyl-L-cysteine) 是 New Delhi metallo-beta-lactamase-1 (NDM-1) 的抑制剂 (IC50 = 1000 μM)。 | |||
T6625 |
Ozagrel hydrochloride
Ozagrel HCl,盐酸奥扎格雷,OKY-046 HCl |
Thrombin; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Proteases/Proteasome |
Ozagrel hydrochloride (OKY-046 HCl) 是一种选择性血栓素 A(2) 合成酶抑制剂,用于改善术后脑血管收缩和伴随的脑缺血。它是一种抗血小板剂,可选择性抑制人血小板聚集,IC50为 53.12 μM。 | |||
T4190 |
Ticlopidine
PCR 5332,Ticlid,噻氯匹定 |
ATPase; Adiponectin receptor | GPCR/G Protein; Membrane transporter/Ion channel |
Ticlopidine (PCR 5332) 是抗血栓前药。它是CYP2C19人肝细胞色素的抑制剂,抑制 CYP2C9 及 CYP3A4。他是变构CD39的非竞争性抑制剂,能够阻断 NTPDase 同工酶,对NTPDase2和NTPDase3的IC50分别为 170 µM 和 149 µM。 | |||
T8719 |
SC99
|
Apoptosis; JAK; STAT | Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells |
SC99 是一种口服有效选择性STAT3抑制剂,靶向 JAK2-STAT3 途径,抑制血小板活化和聚集,有抗骨髓瘤和抗血栓活性。它结合在 JAK2 的 ATP 结合袋中,抑制 JAK2 和 STAT3 的磷酸化。 | |||
T0230 |
Prasugrel
LY640315,CS-747,普拉格雷,PCR 4099 |
P2Y Receptor | GPCR/G Protein; Neuroscience |
Prasugrel (CS-747) 是一种噻吩吡啶和前药,是一种可口服的 P2Y12受体拮抗剂,抑制 ADP 诱导的血小板聚集,用于预防急性冠状动脉综合征患者的血栓形成、不稳定型心绞痛和心肌梗塞,以及接受经皮冠状动脉介入治疗的患者。 | |||
T1893 |
Parmodulin 2
ML 161 |
Protease-activated Receptor | GPCR/G Protein |
Parmodulin 2 (ML 161) 是一种蛋白酶激活受体 1(PAR1) 变构抑制剂,IC50为 0.26 μM。它是蛋白酶激活受体 1 (PAR1) 介导的血小板活化的抑制剂,可以抑制体外血小板聚集和体内血小板血栓形成。 | |||
T16164 |
MY-5445
N-(3-chlorophenyl)-4-phenylphthalazin-1-amine |
PDE | Metabolism |
MY-5445 (N-(3-chlorophenyl)-4-phenylphthalazin-1-amine) 是特异性的 cGMP 磷酸二酯酶 PDE5抑制剂,其 Ki=1.3 μM。它是一种 ABCG2转运蛋白调节剂,具有抗增殖活性。它能抑制人血小板凝集。 | |||
T2569 |
Chlorotrianisene
tris(p-methoxyphenyl)chloroethylene,氯丁烯二烯,CTA,tri-p-anisylchloroethylene,氯烯雌醚,TACE |
Estrogen Receptor/ERR; Estrogen/progestogen Receptor; COX | Endocrinology/Hormones; Immunology/Inflammation; Neuroscience |
Chlorotrianisene (tri-p-anisylchloroethylene) 是长效、可口服、亲脂性高的合成三苯乙烯 (TPE) 衍生物和选择性雌激素受体调节剂,有雌激素活性,也有抗雌激素活性。它还有效抑制COX-1并抑制全血中的血小板聚集。 | |||
T0182L |
Clopidogrel hydrogen sulfate
硫酸氢氯吡格雷,(S)-(+)-Clopidogrel hydrogen sulfate,(S)-(+)-Clopidogrel bisulfate,SR-25990C,Clopidogrel,硫酸氯吡格雷 |
P450; P2Y Receptor | GPCR/G Protein; Metabolism; Neuroscience |
Clopidogrel hydrogen sulfate ((S)-(+)-Clopidogrel bisulfate) 是一种抗血小板药物,可防止血栓形成。它抑制 CYP2B6和 CYP2C19,IC50分别为 18.2 和 524 nM。 它是一种选择性的高亲和力 P2Y12 受体拮抗剂,可抑制纤维蛋白原与血小板的结合以及血小板的粘附和聚集。 | |||
T6952 |
Prasugrel Hydrochloride
LY 640315,PCR 4099 (hydrochloride),盐酸普拉格雷,Effient Hydrochloride,LY 640315 Hydrochloride,Prasugrel HCl |
P2Y Receptor | GPCR/G Protein; Neuroscience |
Prasugrel Hydrochloride (LY 640315 Hydrochloride) 是一种噻吩吡啶和前药,是一种可口服的P2Y12受体拮抗剂,抑制 ADP 诱导的血小板聚集,用于预防急性冠状动脉综合征患者的血栓形成、不稳定型心绞痛和心肌梗塞,以及接受经皮冠状动脉介入治疗的患者。 | |||
T15757 |
Limaprost
17α,20-dimethyl-δ2-PGE1,利马前列素,OP1206,ONO1206 |
PGE Synthase | Immunology/Inflammation |
Limaprost (17α,20-dimethyl-δ2-PGE1) 是PGE1类似物,也是口服具有活性的血管舒张剂。它能够增加血流量以及减少血小板聚集。它具有抗心绞痛的功能,可用于疼痛的缓解,以及用于研究缺血性症状。 | |||
T1618 |
Dipyridamole
Persantin,Dypyridamole,Dipyridamol,双嘧达莫,NSC-515776,Dipyudamine |
PDE | Metabolism |
Dipyridamole (Persantin) 是一种磷酸二酯酶抑制剂,能阻断红细胞和血管内皮细胞对腺苷的吸收和代谢。 | |||
T8575 |
ENFENAMIC ACID
|
Platelet aggregation | Others |
Enfenamic acid 是一种能够抑制伤口愈合的非甾体抗炎药。 | |||
T3608 |
Carbasalate calcium
Rheomin,Omegin,Alcacyl,Iromin,卡巴匹林钙,Solupsan,Carbasalate Calcium |
Platelet aggregation | Others |
Carbasalate calcium (Rheomin) 是抗炎和解热剂,可用于研究疼痛的缓解。 | |||
T0362 |
Ticlopidine hydrochloride
Ticlodone,Ticlopidine HCl,Ticlodix,盐酸噻氯匹定 |
Adenosine Receptor | GPCR/G Protein; Neuroscience |
Ticlopidine hydrochloride (Ticlodix) 是一种 ADP 受体抑制剂,对血小板凝集的IC50为2 μM。 | |||
T31213 |
Dazmegrel
UK-38,485,UK 38485,UK 38,485,UK38,485,UK-38485 |
PPAR | DNA Damage/DNA Repair; Metabolism |
Dazmegrel (UK 38,485) 是一种强效特异性血栓素 A2(TXA2)合成酶抑制剂,可用于预防正常妊娠中全血小板聚集增加。 | |||
T15577 |
Indobufen
Ibustrin,吲哚布芬 |
COX | Immunology/Inflammation; Neuroscience |
Indobufen (Ibustrin) 是一种血小板聚集抑制剂,是下调单核细胞中的组织因子,可逆抑制血小板环氧合酶 (Cox) 的活性和血栓素 A2 (TxA2) 的合成。 | |||
T25635 |
Lateritin
Bassiatin |
Acyltransferase | Metabolism |
Lateritin (Bassiatin) 是一种酰基辅酶 A,是胆固醇酰基转移酶 (ACAT) 抑制剂和来自赤霉属菌丝饼的血小板聚集抑制剂。 Bassiatin 是 (3S,6R) 异构体。 | |||
T9887 |
ethyl 1-[(4-cyanobenzyl)oxy]-2-(3-cyanophenyl)-4-methyl-1H-imidazole-5-carboxylate
|
Platelet aggregation | Others |
ethyl 1-[(4-cyanobenzyl)oxy]-2-(3-cyanophenyl)-4-methyl-1H-imidazole-5-carboxylate 是一种血小板聚集抑制剂。 | |||
T12808 |
S-Nitroso-N-acetyl-DL-penicillamine
N-乙酰基-3-(硫代亚硝基)-DL-缬氨酸,SNAP |
NO Synthase | Immunology/Inflammation |
S-Nitroso-N-acetyl-DL-penicillamine (SNAP) 是一种稳定的血小板聚集抑制剂,是一氧化氮的供体。 | |||
T10502 |
Benzcyclane
苄环庚烷,Benzcyclan,Bencyclane |
Others; Platelet aggregation | Others |
Benzcyclane (Benzcyclan) 是一种血小板聚集抑制剂,也是一种血管扩张剂,可用于多种外周循环障碍。 | |||
T24567 |
Octimibate
Octimibato |
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Octimibate (Octimibato) 是一种非前列腺素类血小板聚集抑制剂和环前列腺素激动剂。Octimibate 可用于治疗心血管疾病,可用于研究动脉粥样硬化和血栓形成。 | |||
T29097 |
VAS 3947
VA-S3947,VA S3947,VAS3947 |
Apoptosis; NADPH-oxidase | Apoptosis; Immunology/Inflammation |
VAS 3947 是一种特异的 NADPH 氧化酶 (NOX) 抑制剂。VAS 3947具有强大的抗血小板作用, 通过 UPR 激活,主要由于蛋白质聚集和错误折叠,独立于抗 NOX 活性诱导细胞凋亡。 | |||
T15130 |
Dilazep dihydrochloride
|
Others | Others |
Dilazep dihydrochloride 是一种腺苷摄取的抑制剂。它可抑制缺血性损伤,血小板聚集和核苷的膜转运。它能够增强腺苷的作用,进而具有脑和冠状血管舒张作用。 | |||
T0179 |
Ticagrelor
替格瑞洛,替卡格雷,AR-C 126532XX,AZD6140 |
P450; P2Y Receptor | GPCR/G Protein; Metabolism; Neuroscience |
Ticagrelor (AR-C 126532XX) (AZD6140) 是可逆的,可口服的 P2Y12受体拮抗剂,可抑制血小板聚集。 | |||
T6040 |
Aloxistatin
E64d,Loxistatin,阿洛司他丁,E64c ethyl ester |
SARS-CoV; Cysteine Protease | Microbiology/Virology; Proteases/Proteasome |
Aloxistatin (E64d) 是一种不可逆的、可透过膜的溶酶体和细胞溶质半胱氨酸蛋白酶抑制剂,能够抑制完整血小板中的钙蛋白酶活性。它是一种半胱氨酸蛋白酶抑制剂,具有血小板聚集抑制活性。 | |||
T76844 |
Abciximab
C7E3 |
Integrin | Cytoskeletal Signaling |
Abciximab (C7E3) 是一种小鼠/人嵌合单克隆抗体,是一种有效的糖蛋白 IIb/IIIa (glycoprotein IIb/IIIa) 抑制剂。 Abciximab 具有抗血小板聚集和白细胞粘附的作用,通过与糖蛋白 IIb/IIIa、vitronectin 和 Mac-1 受体结合发挥作用。 | |||
T17039 |
Terbogrel
BIBV 308SE |
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Terbogrel 是一种可口服的 、具有选择性 thromboxane A2 受体拮抗剂(IC50 约为 10 nM),是一种 thromboxane A2 synthase 抑制剂(IC50 约为 10 nM)。Terbogrel 是一种抗血小板化合物,可抑制血小板聚集,是预防血栓的潜在化合物。 | |||
T23899 |
Cloricromen
O=C(OCC)COC1=CC=C(C(O2)=C1Cl)C(C)=C(CCN(CC)CC)C2=O |
||
Cloricromen is an inhibitor of platelet aggregation. | |||
T68995 | AQ 1994 | ||
AQ 1994 is a platelet aggregation inhibitor. | |||
T71367 |
OM-4842
|
||
OM-4842 is a platelet aggregation inhibitor from Streptomyces. | |||
T68996 |
AQ 1989
|
||
AQ 1989 is a platelet aggregation inhibitor. | |||
T68902 |
Talosalate
|
||
Talosalate is an inhibitor of blood platelet aggregation. | |||
T68832 | Itazigrel | ||
Itazigrel is a platelet aggregation inhibitor. | |||
T69154 | AY-16804 | ||
AY-16804 is an inhibitor of platelet aggregation. | |||
T11629 | Ifenprodil glucuronide | Others | Others |
Ifenprodil glucuronide, a derivative of Ifenprodil, is a vasodilator and an inhibitor of platelet aggregation. In contrast to Ifenprodil, Ifenprodil glucuronide does not affect platelet aggregation nor arterial contraction. | |||
T27408 |
Gea 3162
Gea3162,Gea-3162 |
||
Gea 3162 is a potent inhibitor of ADP-induced platelet aggregation in platelet rich plasma (PRP). GEA 3162 stimulates cGMP production in granulocytes, platelets, and polymorphonuclear leukocytes. | |||
T25364 |
Efegatran
LY 294468,LY294468,LY-294468 |
||
Efegatran is a hematologic agent and platelet aggregation inhibitor. | |||
T68433 |
Clinprost
|
||
Clinprost is a Vasodilator (peripheral), Platelet aggregation inhibitor, and Prostaglandin I2 receptor agonist | |||
T26072 | Rhazimine | ||
Rhazimine is an indole alkaloid. It is a dual inhibitor of arachidonic acid metabolism and platelet activating factor-induced platelet aggregation. | |||
T15238 |
Epoprostenol sodium
Prostaglandin I2 sodium salt,Prostacyclin sodium salt,Flolan |
Others | Others |
Epoprostenol sodium is a potent inhibitor of platelet aggregation used in pulmonary hypertension and transplantation. | |||
T24745 |
RUC-1
RUC1 |
||
RUC-1 is an αIIbβ3-selective ADP-induced platelet aggregation inhibitor. | |||
T68751 | Hoe 892 | ||
Hoe 892 is a stable thia-thimo-analogue of prostacyclin and acts as a platelet aggregation inhibitor. | |||
T68251 | Domipizone | ||
Domipizone is a platelet aggregation inhibitor, cardiotonic and vasodilator. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6S0139 |
Neobavaisoflavone
|
Apoptosis; DNA/RNA Synthesis | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Neobavaisoflavone 是一种从Psoralea corylifolia 的种子中分离出来的类黄酮。它具有抗炎,抗癌和抗氧化的作用。它在中至高浓度下可抑制 DNA 聚合酶,也可抑制血小板聚集。 | |||
T3781 |
Jujuboside B
酸枣仁皂苷 B,酸枣仁皂苷B |
Others | Others |
Jujuboside B 是一种提取自Zizyphus jujuba 中的活性成分,对血小板聚集具有抑制作用。 | |||
T3S1591 |
Notoginsenoside Fc
三七皂苷 FC,三七皂苷Fc |
Others; Autophagy | Autophagy; Others |
Notoginsenoside Fc 是从三七叶中分离得到的原卟啉二醇型皂苷,可通过促进自噬促进糖尿病大鼠血管损伤后的内皮细胞再生,具有抗血小板聚集的作用。 | |||
T0853 |
Adenosine
腺苷,D-Adenosine,Adenine riboside |
Apoptosis; Nucleoside Antimetabolite/Analog; Endogenous Metabolite; Autophagy | Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism |
Adenosine (D-Adenosine) 是一种核糖核苷,由与核糖结合的腺嘌呤组成,具有血管扩张、抗心律失常和镇痛作用。 | |||
TN2244 |
Sulfuretin
硫黄菊素 |
NF-κB; Autophagy | Autophagy; NF-κB |
Sulfuretin 是竞争性单酚酶和二酚酶活性抑制剂,IC50=13.64 μM。它通过抑制NF-κB 通路来抑制炎症反应。 它可用于过敏性气道炎症的研究。它减少氧化应激、血小板聚集和诱变。 | |||
T1626 |
Prostaglandin E1
前列地尔,PGE1,列腺素E1,Alprostadil |
Endogenous Metabolite; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Metabolism |
Prostaglandin E1 (Alprostadil) 是一种前列腺素受体配体,对小鼠 EP1、EP2、EP3、EP4和 IP 的 Ki 值分别为 36、10、1.1、2.1 和 33 nM。它诱导血管舒张并抑制血小板聚集,可作为血管扩张剂用于外周血管疾病的研究。 | |||
TN4222 |
Homoeriodictyol 7-O-β-D-glucoside
高圣草素-7-O-Β-D-葡萄糖苷,Homoeriodictyol 7-O-glucoside |
Others; Platelet aggregation | Others |
Homoeriodictyol 7-O-β-D-glucoside (Homoeriodictyol 7-O-glucoside) 是 Viscum coloratum(Kom.)Nakai 的天然产物。Homoeriodictyol 7-O-β-D-glucoside 是血小板活化因子 (PAF) 的拮抗剂。 | |||
TN6924 |
Anhydrosafflor yellow B
(2S,3S)-6,7-dihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-2-[(1S,2R,3R)-1,2,3,4-tetrahydroxybutyl]-3-{2,3,4-trihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-6-oxo-3-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]cyclohexa-1,4-dien-1,脱水红花黄色素B,AHSYB |
Others | Others |
Anhydrosafflor yellow B ((2S,3S)-6,7-dihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-2-[(1S,2R,3R)-1,2,3,4-tetrahydroxybutyl]-3-{2,3,4-trihydroxy-5-[(2E)-3-(4-hydroxyphenyl)prop-2-enoyl]-6-oxo-3-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]cyclohexa-1,4-dien-1) 是从红花中分离出来的,可抑制 ADP 诱导的血小板聚集,在体外表现出显着的抗氧化作用,并对 H2O2 诱导的细胞毒性具有一定的活性。 | |||
T28551 |
Ro 09-0680
Ro 09 0680,Ro-09-0680 |
||
Ro 09-0680 is an inhibitor of platelet aggregation. | |||
T12164 |
N6-(4-Hydroxybenzyl)adenosine
Para-topolin riboside,N6-羟苄腺苷 |
P2Y Receptor | GPCR/G Protein; Neuroscience |
N6-(4-Hydroxybenzyl)adenosine (Para-topolin riboside) 是一种血小板聚集抑制剂。 | |||
T3734 |
3',4'-Dihydroxyacetophenone
二羟基苯乙酮,Qingxintong,4-Acetylpyrocatechol |
Tyrosinase; Platelet aggregation | Others; Proteases/Proteasome |
3',4'-Dihydroxyacetophenone (Qingxintong) 是一种血管活性物质和抗氧化剂,可从Picea Schrenkiana 中分离得到,能抑制酪氨酸酶,其IC50=10 μM。 | |||
TN1254 |
3'-Methoxydaidzein
3'-甲氧基大豆苷元 |
Sodium Channel | Membrane transporter/Ion channel |
3'-Methoxydaidzein 是一种异黄酮和 Sodium Channel 双重抑制剂。3'-Methoxydaidzein 对NaV1.7、NaV1.8 和 NaV1.3有抑制作用,IC50 分别为 181 nM、397 nM 和 505 nM。 3'-Methoxydaidzein 对胶原诱导的血小板聚集具有特异性,IC50值分别为12.3和61.5µM。。3'-Methoxydaidzein 通过抑制电压门控钠通道发挥镇痛作用。 3'-Methoxydaidzein 具有抗氧化活性和抗血小板聚集活性。 | |||
T3S0645 |
N-trans-Feruloyltyramine
Feruloyltyramine,N-Feruloyltyramine,Moupinamide,N-反式阿魏酰酪胺 |
Others; COX | Immunology/Inflammation; Neuroscience; Others |
N-trans-Feruloyltyramine (Feruloyltyramine) 是从大麻中分离得到的一种生物碱,是COX1和COX2的抑制剂,具有抗氧化和抗炎活性。 | |||
T17273 |
YM-254890
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Others | Others |
YM-254890 inhibits platelet aggregation induced by ADP by blocking the P2Y1 signal transduction pathway (IC50: below 0.6 μM). YM-254890 is a selective Gαq/11 protein inhibitor. YM-254890 displays no inhibition of other G protein subtypes. | |||
T82003 | Juniferdin | ||
Juniferdin是一种抑制Protein disulfide isomerase (PDI),IC50为3.5 μM,旨在阻断HIV传播的化合物。此外,Juniferdin展现出细胞毒性并能抑制血小板聚集。 | |||
T36295 | Echistatin TFA | ||
Echistatin TFA, the smallest active RGD protein belonging to the family of disintegrins that are derived from snake venoms, is a potent inhibitor of platelet aggregation. Echistatin is a potent inhibitor of bone resorption in culture. Echistatin is a potent antagonist of αIIbβ3, αvβ3 and α5β1[1][2][3][4]. [1]. J Musial, et al. Inhibition of platelet adhesion to surfaces of extracorporeal circuits by disintegrins. RGD-containing peptides from viper venoms. Circulation. 1990 Jul;82(1):261-73.[2]. ... | |||
T64246 | Cinchonine monohydrochloride hydrate | ||
Cinchonine ((8R,9S)-Cinchonine) monohydrochloride hydrate 是一种天然的、有效的抗疟剂,也是一种人血小板聚集的抑制剂。Cinchonine monohydrochloride hydrate 能够激活内质网应激,诱导的人肝癌细胞凋亡,并可抑制脂肪的生成。 | |||
TN5221 | (-)-Variabilin | ||
Variabilin, a novel inhibitor of human platelet aggregation, it is a potent RGD (Arg-Gly-Asp)-containing antagonist of the fibrinogen receptor glycoprotein IIb-IIIa (GPIIb-IIIa; αIIbβ3) and the vitronectin receptor αvβ3.Variabilin is also an antimicrobial furanosesterterpene. Variabilin is an inhibitor of human secretory and cytosolic phospholipase A2 (PLA2) activities that controls eicosanoid production in vitro and in vivo, inhibits neutrophil degranulation and superoxide generation in vitro a... | |||
T72916 |
Justicidin B
爵床脂素B |
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Justicidin B是一种高效的抗癌木脂素及促凋亡剂,同时具备显著的骨吸收抑制作用,并展现出强大的抗病毒、杀真菌和抗原虫能力。此外,Justicidin B能显着抑制血小板聚集。 |